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Escalation Regimen for LAMICTAL XR in Patients Aged 13 Years and OlderIn Patients NOT TAKING Carbamazepine, Phenytoin, Phenobarbital, Primidone,In Patients TAKING Carbamazepine, Phenytoin, Phenobarbital, or PrimidoneConversion from Adjunctive Therapy with Carbamazepine, Phenytoin, Phenobarbital, or Primidone to Monotherapy with LAMICTAL XRConversion from Adjunctive Therapy with Valproate to Monotherapy with LAMICTAL XRTable 2. Avoid use with other CNS depressants at bedtime; avoid use with alcohol.May interfere with some rapid urine drug screens, particularly phencyclidine (false-positives).Percentages reported in adults on monotherapy for epilepsy or bipolar disorder.Cardiovascular: Chest pain (2% to 5%), peripheral edema (2% to 5%), edema (1% to 5%)Central nervous system: Insomnia (5% to 10%), drowsiness (9%), fatigue (8%), dizziness (7%), ataxia (2% to 7%), anxiety (5%), pain (5%), irritability (2% to 5%), suicidal ideation (2% to 5%), abnormal dreams (1% to 5%), abnormality in thinking (1% to 5%), agitation (1% to 5%), amnesia (1% to 5%), depression (1% to 5%), emotional lability (1% to 5%), hypoesthesia (1% to 5%), migraine (1% to 5%), neurologic abnormality (dyspraxia) (1% to 5%), hyperreflexia (>2% to <5%), hyporeflexia (>2% to <5%), confusion (≥1%), paresthesia (≥1%)Dermatologic: Skin rash (nonserious: 7%; requiring hospitalization: ≤1%), contact dermatitis (2% to 5%), diaphoresis (2% to 5%), xeroderma (2% to 5%)Endocrine & metabolic: Increased libido (2% to 5%), weight loss (2% to 5%), weight gain (1% to 5%)Gastrointestinal: Vomiting (5% to 9%), dyspepsia (7%), abdominal pain (6%), xerostomia (2% to 6%), constipation (5%), anorexia (2% to 5%), peptic ulcer (2% to 5%), flatulence (1% to 5%)Genitourinary: Dysmenorrhea (2% to 5%), urinary frequency (1% to 5%)Hematologic & oncologic: Rectal hemorrhage (2% to 5%)Neuromuscular & skeletal: Back pain (8%), asthenia (2% to 5%), arthralgia (1% to 5%), myalgia (1% to 5%), neck pain (1% to 5%)Ophthalmic: Nystagmus disorder (2% to 5%), visual disturbance (2% to 5%), amblyopia (≥1%)Respiratory: Rhinitis (7%), cough (5%), pharyngitis (5%), bronchitis (2% to 5%), dyspnea (2% to 5%), epistaxis (2% to 5%), sinusitis (1% to 5%), nasopharyngitis (≥3%), upper respiratory tract infection (≥3%)Hematologic & oncologic: Natural killer cell count increased (hemophagocytic lymphohistiocytosis)<1%, postmarketing and/or case reports (any indication): Abnormal hepatic function tests, abnormal lacrimation, accommodation disturbance, acne vulgaris, acute renal failure, ageusia, aggressive behavior, agranulocytosis, akathisia, alcohol intolerance, alopecia, altered sense of smell, amyotrophy, anemia, angioedema, anorgasmia, apathy, aphasia, aplastic anemia, apnea, arthritis, aseptic meningitis, blepharoptosis, breast abscess, breast neoplasm, bursitis, central nervous system depression, chills, choreoathetosis, conjunctivitis, cystitis, deafness, decreased fibrin, decreased libido, decreased serum fibrinogen, delirium, delusion, depersonalization, dermatitis (exfoliative, fungal), drug reaction with eosinophilia and systemic symptoms syndrome, dry eye syndrome, dysarthria, dysgeusia, dyskinesia, dysphagia, dysphoria, dystonia, dysuria, ecchymosis, ejaculatory disorder, eosinophilia, epididymitis, eructation, erythema multiforme, erythema of skin, esophagitis, euphoria, exacerbation of Parkinson disease, extrapyramidal reaction, flushing, gastric ulcer, gastritis, gastrointestinal hemorrhage, gingival hemorrhage, gingival hyperplasia, gingivitis, glossitis, goiter, hallucination, heavy menstrual bleeding, hematemesis, hematuria, hemiplegia, hemolytic anemia, hemorrhagic colitis, hepatitis, hepatotoxicity (idiosyncratic) (Chalasani 2014), herpes zoster infection, hiccups, hirsutism, hostility, hot flash, hyperalgesia, hyperbilirubinemia, hyperesthesia, hyperglycemia, hyperkinetic muscle activity, hypersensitivity reaction, hypertension, hypertonia, hyperventilation, hypogammaglobulinemia, hypokinesia, hypothyroidism, hypotonia, immunosuppression (progressive), impotence, increased appetite, increased gamma-glutamyl transferase, increased serum alkaline phosphatase, increased serum alanine aminotransferase, increased serum aspartate aminotransferase, increased serum creatinine, iron deficiency anemia, lactation, leukocytosis, leukoderma, leukopenia, lower limb cramp, lupus-like syndrome, lymphadenopathy, lymphocytosis, macrocytic anemia, maculopapular rash, malaise, manic depressive reaction, melena, memory impairment, movement disorder, multiorgan failure, muscle spasm, myasthenia, myoclonus, neuralgia, neutropenia, nocturia, oral mucosa ulcer, orthostatic hypotension, oscillopsia, otalgia, palpitations, pancreatitis, pancytopenia, panic attack, paralysis, paranoid ideation, pathological fracture, peripheral neuritis, personality disorder, petechia, petechial rash, photophobia, polyuria, pruritus, psychoneurosis, psychosis, pure red cell aplasia, pustular rash, racing mind, renal pain, rhabdomyolysis, sialorrhea, skin discoloration, sleep disorder, status epilepticus, Stevens-Johnson syndrome, stomatitis, strabismus, stupor, suicidal tendencies, syncope, tachycardia, tendinous contracture, thrombocytopenia, tic disorder, tinnitus, tongue edema, tonic clonic epilepsy (exacerbation), toxic epidermal necrolysis, twitching, urinary incontinence, urinary retention, urinary urgency, urticaria, uveitis, vasculitis, vasodilation, vesiculobullous dermatitis, visual field defect, withdrawal syndrome (seizures with abrupt withdrawal), yawningLamotrigine can cause serious rashes requiring hospitalization and discontinuation of treatment.

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